full agonist造句

• Such adverse effects appear to be less problematic with bretazenil than full agonists.
• It acts as a receptor full agonist with a long duration of action.
• Repinotan HCI ( BAYx3702 ) acts as a highly selective 5-HT1A receptor full agonist.
• In a study of monkeys bretazenil has been found to antagonise the effects of full agonist benzodiazepines.
• It was one of the first major 5-HT 1A receptor full agonists to be discovered.
• It is a potent CB 1 full agonist with a K i of 1.16 nM.
• The compound is equipotent at ER? and ER?, and acts as a full agonist of ER?.
• Primarily, it a full agonist on the H 1 receptors located on blood vessels in the inner ear.
• The RPE can be used to define full agonists for ER, between 80 % and 100 % relative proliferation.
• When the piperidine ring of raloxifene is replaced by cyclohexane, the ligand loses antiestrogenic properties and becomes a full agonist.
• "' LY-293284 "'is a research chemical developed by the pharmaceutical company receptor full agonist.
• It behaves as a full agonist at the D 1 protomer and a high-affinity partial agonist at the D 2 protomer.
• Flurazepam is a unique benzodiazepine in that it is a partial agonist of benzodiazepine receptors whereas other benzodiazepines are full agonists of benzodiazepine receptors.
• Another study found that bretazenil acted as an antagonist provoking withdrawal symptoms in monkeys who were physically dependent on the full agonist benzodiazepine triazolam.
• Compared to THC, which is a partial agonist at CB 1 receptors, JWH-018, and many synthetic cannabinoids, are full agonists.
• It is the only selective full agonist for the ? adrenergic receptors known to date and has been used to study their function in scientific research.
• Partial agonists ( such as buspirone, aripiprazole, buprenorphine, or efficacy at the receptor relative to a full agonist, even at maximal receptor occupancy.
• It is a partial agonist at ?1-, ?2-and ?5-containing GABAA receptors and a full agonist at receptors containing an ?3 subunit.
• Methamphetamine has been identified as a potent full agonist of firing rate of neurons through direct activation of G protein-coupled inwardly-rectifying potassium channels.
• "' Dinoxyline "'is a synthetic compound developed for scientific research, which acts as a potent full agonist at all five dopamine receptor subtypes.